{"id":2087,"date":"2024-03-19T17:55:16","date_gmt":"2024-03-19T15:55:16","guid":{"rendered":"https:\/\/sweetdropcbd.com\/?p=2087"},"modified":"2024-03-19T17:55:59","modified_gmt":"2024-03-19T15:55:59","slug":"medicininiai-kanapiu-naudojimo-aspektai","status":"publish","type":"post","link":"https:\/\/sweetdropcbd.com\/lt\/medicininiai-kanapiu-naudojimo-aspektai\/","title":{"rendered":"Medicininiai Kanapi\u0173 Naudojimo Aspektai"},"content":{"rendered":"<p>Kanap\u0117s, moksli\u0161kai vadinamos Cannabis sativa L., Kinijoje medicininiais tikslais naudojamos jau daugiau kaip 4000 met\u0173. Seniausias u\u017efiksuotas medicininis kanapi\u0173 naudojimas priskiriamas legendiniam Kinijos imperatoriui \u0160en Nungui, kuris, kaip manoma, gyveno <a href=\"https:\/\/sweetdropcbd.com\/lt\/apie-mus\/\">apie<\/a> 2700 m. pr. m. e. Kanapi\u0173 naudojimas medicinoje buvo u\u017efiksuotas Shen Nung Pen-ts&#8217;ao Ching, II a. kin\u0173 vaista\u017eoli\u0173 gydymo knygoje, kurioje kalbama apie plat\u0173 spektr\u0105 negalavim\u0173 \u2013 nuo menstruacij\u0173 iki kognityvini\u0173 sutrikim\u0173. I\u0161 prad\u017ei\u0173 kinai vaistams pirmiausia naudojo kanapi\u0173 s\u0117klas. Vaistinis augalo vartojimas i\u0161plito \u012f Indij\u0105, Persij\u0105 ir Asirij\u0105, o v\u0117liau paplito Artimuosiuose Rytuose, Afrikoje, Europoje ir galiausiai Jungtin\u0117se Amerikos Valstijose.<\/p>\n<p>XIX a. Williamas B. O&#8217;Shaughnessy, tarnav\u0119s Indijoje, pristat\u0117 C. sativa \u012f Anglij\u0105. 1839 m. jis i\u0161leido knyg\u0105 &#8222;On Preparations of the Indian Hemp or Gunjah\u201d (&#8222;<a href=\"https:\/\/sweetdropcbd.com\/lt\/apie-mus\/\">Apie<\/a> indi\u0161k\u0173 kanapi\u0173 arba gunjah preparatus\u201d), kurioje i\u0161samiai apra\u0161\u0117 s\u0117kmingus eksperimentus su \u017emon\u0117mis, ypa\u010d su kanapi\u0173 preparatais, skirtais raumen\u0173 spazmams, reumatui ir traukuli\u0173 priepuoliams gydyti. V\u0117liau, XIX a. antroje pus\u0117je ir XX a. prad\u017eioje, Europoje ir Jungtin\u0117se Amerikos Valstijose pasirod\u0117 daug mokslini\u0173 straipsni\u0173 <a href=\"https:\/\/sweetdropcbd.com\/lt\/apie-mus\/\">apie<\/a> kanapi\u0173 gydom\u0105j\u0105 vert\u0119.<\/p>\n<p>Kanap\u0117s yra keli\u0173 r\u016b\u0161i\u0173: Cannabis sativa, Cannabis indica ir Cannabis ruderalis. Kanapi\u0173 r\u016b\u0161yse nustatyta daugiau kaip 500 jungini\u0173, \u012fskaitant ma\u017edaug 100 kanabinoid\u0173, pasi\u017eymin\u010di\u0173 21 anglies terpenofenolio strukt\u016bra. I\u0161 \u0161i\u0173 jungini\u0173 labiausiai paplit\u0119 tetrahidrokanabinolis (THC), sukeliantis psichoaktyv\u0173j\u012f poveik\u012f, ir kanabidiolis (<a href=\"https:\/\/sweetdropcbd.com\/lt\/kodel-sweet-drop-cbd\/\">CBD<\/a>), kuris neturi psichoaktyvumo.<\/p>\n<p>Fitokanabinoidai yra kanabinoidai, kuriuos gamina kanap\u0117s augalas, ir juose nustatyta daugiau kaip 100 nat\u016braliai randam\u0173 chemini\u0173 med\u017eiag\u0173. Be THC ir <a href=\"https:\/\/sweetdropcbd.com\/product\/sweet-drop-5-cbd-oil-500-mg-10ml\/\">CBD<\/a>, gausu terpen\u0173 ir flavonoid\u0173. THC sukelia psichoaktyv\u0173j\u012f poveik\u012f, o <a href=\"https:\/\/sweetdropcbd.com\/lt\/kodel-sweet-drop-cbd\/\">CBD<\/a> n\u0117ra psichotropinis. Pastaruoju metu legalizavus kanapes, spar\u010diai i\u0161augo medicininis kanapi\u0173 ir j\u0173 produkt\u0173 vartojimas, o tai paskatino per\u017ei\u016br\u0117ti j\u0173 veikimo principus ir farmakokinetik\u0105.<\/p>\n<h4><strong>Veikimo principai<\/strong><\/h4>\n<p>Kanabinoid\u0173 poveikio supratimui svarbus etapas buvo endokanabinoid\u0173 sistemos (ECS) nustatymas. THC ir <a href=\"https:\/\/sweetdropcbd.com\/lt\/kodel-sweet-drop-cbd\/\">CBD<\/a> buvo pagrindiniai veiksniai, pad\u0117j\u0119 atrasti ECS signal\u0173 kelius. THC s\u0105veikauja su 1 tipo kanabinoid\u0173 receptoriais (CB1), kurie daugiausia yra centrin\u0117je nerv\u0173 sistemoje, o <a href=\"https:\/\/sweetdropcbd.com\/product\/sweet-drop-15-cbd-oil-1500-mg-10ml\/\">CBD<\/a> s\u0105veikauja su 2 tipo kanabinoid\u0173 receptoriais (CB2), daugiausia i\u0161reik\u0161tais imunin\u0117je sistemoje. Endogeniniai kanabinoidai, tokie kaip anandamidas (AEA) ir 2-arachidonoilglicerolis (2-AG), moduliuoja ECS aktyvum\u0105. Tiek CB1, tiek CB2 receptoriai yra pla\u010diai paplit\u0119 visoje \u0161irdies ir kraujagysli\u0173 sistemoje.<\/p>\n<p>Be s\u0105veikos su CB1 ir CB2 receptoriais, endokanabinoidai ir fitokanabinoidai taip pat s\u0105veikauja su daugeliu kit\u0173 receptori\u0173 ir ferment\u0173, \u012fskaitant \u012fvairius su G baltymais susietus receptorius (GPR55, GPR18, GPR3, GPR6, GPR12), pereinamojo potencialo receptori\u0173 kanalus (TRP vaniljoidai TRPV1- TRPV4, TRP ankyrinas TRPA1, TRP M narys TRPM8), peroksisom\u0173 proliferatori\u0173 aktyvinami receptoriai (PPAR2, PPAR\u03b3), monoamin\u0173 perne\u0161\u0117jai (noradrenalino, dopamino, serotonino 1A receptorius), riebal\u0173 r\u016bg\u0161\u010di\u0173 amid\u0173 hidrolaz\u0117, monoacilglicerolio lipaz\u0117, riebal\u0173 r\u016bg\u0161tis suri\u0161antys transportiniai baltymai, adenozino pusiausvyros nukleozid\u0173 perne\u0161\u0117jai ir glicino receptoriai \u03b11 ir \u03b13.<\/p>\n<p>Atsiranda \u012frodym\u0173, kad endokanabinoid\u0173 funkcija suma\u017e\u0117ja sergant \u012fvairiomis ligomis, pavyzd\u017eiui, migrena, fibromialgija, dirgliosios \u017earnos sindromu, i\u0161s\u0117tine skleroze, diabetine neuropatija, Parkinsono liga ir kt. Pagal endokanabinoid\u0173 tr\u016bkumo teorij\u0105 si\u016bloma, kad toks tr\u016bkumas gali b\u016bti genetin\u0117s, \u012fgimtos ar \u012fgytos kilm\u0117s, atsirad\u0119s d\u0117l su\u017ealojimo ar ligos, tod\u0117l gali atsirasti b\u016bdingi patofiziologiniai sindromai su specifine simptomatika. Fitokanabinoidai, turintys pana\u0161\u0173 poveik\u012f kanabinoid\u0173 receptoriams, gali tapti \u0161i\u0173 sveikatos sutrikim\u0173 gydymo priemon\u0117mis. Sintetiniai kanabinoidai \u2013 tai laboratorijoje pagaminti junginiai, skirti atkartoti endokanabinoid\u0173 arba fitokanabinoid\u0173 strukt\u016br\u0105 ar funkcij\u0105. Dauguma \u0161i\u0173 sintetini\u0173 preparat\u0173 sukurti pagal THC \u2013 nat\u016bral\u0173 kanabinoid\u0105. Jie pasi\u017eymi dideliu giminingumu CB1 receptoriams, kurie siejami su kanapi\u0173 psichoaktyviuoju poveikiu arba kanapi\u0173 &#8222;pakilimu\u201d. Remiantis Europos narkotik\u0173 ir narkomanijos steb\u0117senos centro 2019 m. ataskaitomis, buvo identifikuota ma\u017eiausiai 180 skirting\u0173 sintetini\u0173 kanabinoid\u0173. Paprastai \u0161ie sintetiniai junginiai vartojami r\u016bkant arba koncentruoto skys\u010dio pavidalu. Nepageidaujamas sintetini\u0173 kanabinoid\u0173 poveikis gali b\u016bti \u0161irdies permu\u0161imai, paranoja, stiprus nerimas, pykinimas, v\u0117mimas, sumi\u0161imas, koordinacijos sutrikimas ir traukuliai. \u012edomu tai, kad kai kurie asmenys prane\u0161\u0117, jog net pra\u0117jus savaitei po vartojimo nutraukimo jau\u010dia stipri\u0105 prievart\u0105 ir nuolatin\u012f potrauk\u012f atnaujinti vartojim\u0105, o kiti apra\u0161\u0117 abstinencijos simptomus, tokius kaip galvos skausmas, pykinimas ir v\u0117mimas.<\/p>\n<h4><strong>Farmakokinetika<\/strong><\/h4>\n<p>Kanapi\u0173 med\u017eiag\u0173 kaita priklauso nuo vartojimo b\u016bdo. Vartojant per burn\u0105 THC apykaita vyksta kepenyse, o \u012fkv\u0117pus greitai absorbuojamas per plau\u010dius. <a href=\"https:\/\/sweetdropcbd.com\/product\/sweet-drop-15-cbd-oil-1500-mg-10ml\/\">CBD<\/a>, kaip ir THC, pasi\u017eymi sud\u0117tinga farmakokinetika ir pasi\u017eymi ma\u017eu geriamuoju biologiniu prieinamumu \u012fvairiose r\u016b\u0161yse. Tiek THC, tiek <a href=\"https:\/\/sweetdropcbd.com\/lt\/kodel-sweet-drop-cbd\/\">CBD<\/a> s\u0105veikauja su citochromo P450 fermentais, tod\u0117l gali pakisti \u012fvairi\u0173 vaist\u0173 metabolizmas. Buvo i\u0161reik\u0161tas susir\u016bpinimas d\u0117l THC patekimo per motinos pien\u0105, tod\u0117l pabr\u0117\u017etas atsargumas n\u0117\u0161tumo ir \u017eindymo laikotarpiu.<\/p>\n<p>Apibendrinant galima teigti, kad kanap\u0117s ir j\u0173 sudedamosios dalys turi turting\u0105 istorij\u0105 medicinoje, o j\u0173 terapinis potencialas ir farmakologinis poveikis nuolat tiriami moksliniais tyrimais. Kanapi\u0173 veikimo mechanizm\u0173 ir farmakokinetikos supratimas yra labai svarbus siekiant maksimaliai padidinti j\u0173 medicinin\u0119 naud\u0105 ir kartu suma\u017einti galim\u0105 rizik\u0105.<\/p>\n<p><em>\u0160altinis: https:\/\/www.ncbi.nlm.nih.gov\/pmc\/articles\/PMC8803256\/<\/em><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Kanap\u0117s, moksli\u0161kai vadinamos Cannabis sativa L., Kinijoje medicininiais tikslais naudojamos jau daugiau kaip 4000 met\u0173. Seniausias u\u017efiksuotas medicininis kanapi\u0173 naudojimas priskiriamas legendiniam Kinijos imperatoriui \u0160en Nungui, kuris, kaip manoma, gyveno apie 2700 m. pr. m. e. Kanapi\u0173 naudojimas medicinoje buvo u\u017efiksuotas Shen Nung Pen-ts&#8217;ao Ching, II a. kin\u0173 vaista\u017eoli\u0173 gydymo knygoje, kurioje kalbama apie plat\u0173 [&#8230;]\n","protected":false},"author":1,"featured_media":2088,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[434,438,441],"tags":[446,444,445,442],"class_list":["post-2087","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-cbd-lt","category-cbd-aliejus","category-nepriskirta-kategorijai","tag-cbd","tag-cbd-aliejus","tag-cbd-kanapiu-aliejus","tag-sweet-drop-cbd"],"yoast_head":"<!-- This site is optimized with the Yoast SEO Premium plugin v27.4 (Yoast SEO v27.4) - https:\/\/yoast.com\/product\/yoast-seo-premium-wordpress\/ -->\n<title>Medicininiai Kanapi\u0173 Naudojimo Aspektai - Sweet Drop CBD<\/title>\n<meta name=\"description\" content=\"Su\u017einokite apie kanapi\u0173 (CBD) naudojim\u0105 medicinoje, veikimo mechanizmus. 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