{"id":2669,"date":"2024-03-19T17:55:16","date_gmt":"2024-03-19T15:55:16","guid":{"rendered":"https:\/\/sweetdropcbd.com\/?p=2669"},"modified":"2026-01-30T13:11:41","modified_gmt":"2026-01-30T11:11:41","slug":"kanepju-lietosanas-mediciniskie-aspekti","status":"publish","type":"post","link":"https:\/\/sweetdropcbd.com\/lv\/kanepju-lietosanas-mediciniskie-aspekti\/","title":{"rendered":"Ka\u0146epju lieto\u0161anas medic\u012bniskie aspekti"},"content":{"rendered":"<p><a href=\"https:\/\/sweetdropcbd.com\/lv\/kanabidiols-jauna-alternativa-trauksmes-depresijas-un-psihotisko\/\">Ka\u0146epes<\/a>, zin\u0101tniski paz\u012bstamas k\u0101 <em>Cannabis sativa<\/em> L., \u0136\u012bn\u0101 medic\u012bniskiem nol\u016bkiem tiek izmantotas jau vair\u0101k nek\u0101 4000 gadus. Agr\u0101kais dokument\u0113tais ka\u0146epju \u0101rstnieciskais pielietojums tiek pied\u0113v\u0113ts le\u0123end\u0101rajam \u0137\u012bnie\u0161u imperatoram \u0160e\u0146 Nunam (Shen Nung), kur\u0161, dom\u0101jams, dz\u012bvojis ap 2700. gadu p.m.\u0113. Ka\u0146epju \u0101rstniecisk\u0101 izmanto\u0161ana ir aprakst\u012bta <em>Shen Nung Pen-ts\u2019ao Ching<\/em> \u2014 2. gadsimta \u0137\u012bnie\u0161u \u0101rstniec\u012bbas augu gr\u0101mat\u0101, kur\u0101 apl\u016bkots pla\u0161s kai\u0161u loks, s\u0101kot no menstru\u0101ciju trauc\u0113jumiem l\u012bdz kognit\u012bviem trauc\u0113jumiem. S\u0101kotn\u0113ji \u0137\u012bnie\u0161i medic\u012bn\u0101 galvenok\u0101rt izmantoja ka\u0146epju s\u0113klas. Auga izmanto\u0161ana izplat\u012bj\u0101s uz Indiju, Persiju un As\u012briju, p\u0113c tam uz Tuvajiem Austrumiem, \u0100friku, Eiropu un galu gal\u0101 ar\u012b uz Amerikas Savienotaj\u0101m Valst\u012bm.<\/p>\n<p>19 gadsimt\u0101 Viljams B. O\u2019\u0160o\u0123nesijs (William B. O\u2019Shaughnessy), kur\u0161 dien\u0113ja Indij\u0101, ieviesa <em>C. sativa<\/em> Anglij\u0101. 1839. gad\u0101 vi\u0146\u0161 public\u0113ja darbu <em>On Preparations of the Indian Hemp or Gunjah<\/em>, kur\u0101 aprakst\u012bja savus veiksm\u012bgos eksperimentus ar cilv\u0113kiem, \u012bpa\u0161i ka\u0146epju prepar\u0101tu izmanto\u0161anu musku\u013cu spazmu, reimatisma un krampju l\u0113kmju \u0101rst\u0113\u0161an\u0101. V\u0113l\u0101k, 19. gadsimta otraj\u0101 pus\u0113 un 20. gadsimta s\u0101kum\u0101, Eirop\u0101 un Amerikas Savienotaj\u0101s Valst\u012bs par\u0101d\u012bj\u0101s liels skaits zin\u0101tnisku publik\u0101ciju par ka\u0146epju terapeitisko v\u0113rt\u012bbu.<\/p>\n<p>Ka\u0146epes ir pieejamas vair\u0101k\u0101s sug\u0101s: <em>Cannabis sativa<\/em>, <em>Cannabis indica<\/em> un <em>Cannabis ruderalis<\/em>. Ka\u0146epju sug\u0101s identific\u0113ti vair\u0101k nek\u0101 500 savienojumi, tostarp ap 100 kanabino\u012bdu ar 21 oglek\u013ca terpenofenola strukt\u016bru. No \u0161iem savienojumiem visbie\u017e\u0101k sastopami ir tetrahidrokanabinols (THC), kas izraisa psihoakt\u012bvu iedarb\u012bbu, un kanabidiols (CBD), kam nav psihoakt\u012bvas iedarb\u012bbas.<\/p>\n<p>Fitokanabino\u012bdi ir kanabino\u012bdi, ko ra\u017eo ka\u0146epju augs, un tie ietver vair\u0101k nek\u0101 100 dab\u0101 sastopamu \u0137\u012bmisku vielu. Papildus THC un CBD ka\u0146ep\u0113s ir daudz terp\u0113nu un flavono\u012bdu. THC rada psihoakt\u012bvu iedarb\u012bbu, savuk\u0101rt CBD nav psihotrops. Nesen\u0101 ka\u0146epju legaliz\u0101cija ir veicin\u0101jusi strauju medic\u012bnisk\u0101s ka\u0146epju lieto\u0161anas un to produktu pieaugumu, kas savuk\u0101rt rosin\u0101jis p\u0101rskat\u012bt to darb\u012bbas meh\u0101nismus un farmakokin\u0113tiku.<\/p>\n<p><strong>Darb\u012bbas principi<\/strong><\/p>\n<p>Svar\u012bgs solis kanabino\u012bdu iedarb\u012bbas izpratn\u0113 bija endokanabino\u012bdu sist\u0113mas (ECS) identific\u0113\u0161ana. THC un CBD bija b\u016btiski ECS sign\u0101lce\u013cu atkl\u0101\u0161an\u0101. THC mijiedarbojas ar 1. tipa kanabino\u012bdu receptoriem (CB1), kas p\u0101rsvar\u0101 atrodas centr\u0101laj\u0101 nervu sist\u0113m\u0101, savuk\u0101rt CBD mijiedarbojas ar 2. tipa kanabino\u012bdu receptoriem (CB2), kas p\u0101rsvar\u0101 izteikti im\u016bnsist\u0113m\u0101. Endog\u0113nie kanabino\u012bdi, piem\u0113ram, anandam\u012bds (AEA) un 2-arahidonilglicerols (2-AG), modul\u0113 ECS aktivit\u0101ti. Gan CB1, gan CB2 receptori ir pla\u0161i izplat\u012bti vis\u0101 sirds-asinsvadu sist\u0113m\u0101.<\/p>\n<p>Papildus mijiedarb\u012bbai ar CB1 un CB2 receptoriem endokanabino\u012bdi un fitokanabino\u012bdi mijiedarbojas ar\u012b ar pla\u0161u citu receptoru un enz\u012bmu kl\u0101stu, tostarp da\u017e\u0101diem G olbaltumvielu saist\u012btajiem receptoriem (GPR55, GPR18, GPR3, GPR6, GPR12), p\u0101rejo\u0161\u0101 receptoru potenci\u0101la kan\u0101liem (TRP vanilo\u012bdu TRPV1\u2013TRPV4, TRP ankir\u012bna TRPA1, TRP M apak\u0161grupas TRPM8), peroksisomu proliferatora aktiv\u0113tajiem receptoriem (PPAR2, PPAR\u03b3), monoam\u012bnu transport\u0113t\u0101jiem (noradrenal\u012bna, dopam\u012bna, seroton\u012bna 1A receptoriem), tauksk\u0101bju am\u012bda hidrol\u0101zei, monoacilglicerola lip\u0101zei, tauksk\u0101bju saisto\u0161ajiem transportprote\u012bniem, adenoz\u012bna l\u012bdzsvara nukleoz\u012bdu transport\u0113t\u0101jiem un glic\u012bna receptoriem \u03b11 un \u03b13.<\/p>\n<p>Par\u0101d\u0101s pier\u0101d\u012bjumi, ka endokanabino\u012bdu funkcija ir samazin\u0101ta da\u017e\u0101d\u0101s slim\u012bb\u0101s, piem\u0113ram, migr\u0113n\u0101, fibromial\u0123ij\u0101, kairin\u0101tu zarnu sindrom\u0101, multiplo sklerozi, diab\u0113tisk\u0101 neirop\u0101tij\u0101, Parkinsona slim\u012bb\u0101 u.c. Endokanabino\u012bdu defic\u012bta teorija paredz, ka \u0161\u0101ds defic\u012bts var b\u016bt \u0123en\u0113tisks, iedzimts vai ieg\u016bts traumas vai slim\u012bbas d\u0113\u013c un var izrais\u012bt rakstur\u012bgus patofiziolo\u0123iskus sindromus ar specifisku simptom\u0101tiku. Fitokanabino\u012bdi ar l\u012bdz\u012bgu iedarb\u012bbu uz kanabino\u012bdu receptoriem var sniegt \u0101rst\u0113\u0161anas iesp\u0113jas \u0161iem vesel\u012bbas st\u0101vok\u013ciem. Sint\u0113tiskie kanabino\u012bdi ir laboratorij\u0101 rad\u012bti savienojumi, kas izstr\u0101d\u0101ti, lai atdarin\u0101tu endokanabino\u012bdu vai fitokanabino\u012bdu strukt\u016bru vai funkciju. Liel\u0101k\u0101 da\u013ca \u0161o sint\u0113tisko prepar\u0101tu ir balst\u012bti uz THC \u2014 dabisku kanabino\u012bdu. Tiem ir augsta afinit\u0101te pret CB1 receptoriem, kas saist\u012bti ar ka\u0146epju psihoakt\u012bvo iedarb\u012bbu jeb \u201capreibumu\u201d. Saska\u0146\u0101 ar Eiropas Narkotiku un narkom\u0101nijas uzraudz\u012bbas centra (EMCDDA) 2019. gada zi\u0146ojumiem ir identific\u0113ti vismaz 180 da\u017e\u0101di sint\u0113tiskie kanabino\u012bdi. \u0160os sint\u0113tiskos savienojumus parasti lieto sm\u0113\u0137\u0113jot vai koncentr\u0113ta \u0161\u0137idruma veid\u0101. Sint\u0113tisko kanabino\u012bdu nev\u0113lam\u0101s blakuspar\u0101d\u012bbas var ietvert sirdsl\u0113kmes, paranoju, smagu trauksmi, nelabumu, vem\u0161anu, apjukumu, koordin\u0101cijas trauc\u0113jumus un krampjus. Interesanti, ka da\u017ei indiv\u012bdi ir zi\u0146oju\u0161i par sp\u0113c\u012bgu kompuls\u012bvu tieksmi un notur\u012bgu v\u0113lmi ats\u0101kt lieto\u0161anu pat vienu ned\u0113\u013cu p\u0113c atme\u0161anas, savuk\u0101rt citi ir aprakst\u012bju\u0161i atcel\u0161anas simptomus, piem\u0113ram, galvass\u0101pes, nelabumu un vem\u0161anu.<\/p>\n<p><strong>Farmakokin\u0113tika<\/strong><\/p>\n<p>Ka\u0146epju vielu iedarb\u012bbas at\u0161\u0137ir\u012bbas ir atkar\u012bgas no lieto\u0161anas veida. THC, lietojot iek\u0161\u0137\u012bgi, tiek metaboliz\u0113ts akn\u0101s, bet ieelpojot tas \u0101tri uzs\u016bcas caur plau\u0161\u0101m. CBD, l\u012bdz\u012bgi k\u0101 THC, piem\u012bt sare\u017e\u0123\u012bta farmakokin\u0113tika un zema peror\u0101l\u0101 biopieejam\u012bba da\u017e\u0101d\u0101s sug\u0101s. Gan THC, gan CBD mijiedarbojas ar citohroma P450 enz\u012bmiem, kas var main\u012bt da\u017e\u0101du z\u0101\u013cu metabolismu. Ir paustas ba\u017eas par THC non\u0101k\u0161anu m\u0101tes pien\u0101, t\u0101p\u0113c gr\u016btniec\u012bbas un z\u012bd\u012b\u0161anas laik\u0101 tiek uzsv\u0113rta piesardz\u012bba.<\/p>\n<p>Nosl\u0113gum\u0101 j\u0101secina, ka ka\u0146ep\u0113m un to sast\u0101vda\u013c\u0101m ir bag\u0101ta medic\u012bniska v\u0113sture, un to terapeitiskais potenci\u0101ls un farmakolo\u0123isk\u0101 iedarb\u012bba joproj\u0101m tiek akt\u012bvi p\u0113t\u012bti. Ka\u0146epju darb\u012bbas meh\u0101nismu un farmakokin\u0113tikas izpratne ir b\u016btiska, lai maksim\u0101li palielin\u0101tu to medic\u012bniskos ieguvumus un vienlaikus mazin\u0101tu iesp\u0113jamos riskus.<\/p>\n<p>Avots: <a href=\"https:\/\/www.ncbi.nlm.nih.gov\/pmc\/articles\/PMC8803256\/\">https:\/\/www.ncbi.nlm.nih.gov\/pmc\/articles\/PMC8803256\/<\/a><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Ka\u0146epes, zin\u0101tniski paz\u012bstamas k\u0101 Cannabis sativa L., \u0136\u012bn\u0101 medic\u012bniskiem nol\u016bkiem tiek izmantotas jau vair\u0101k nek\u0101 4000 gadus. Agr\u0101kais dokument\u0113tais ka\u0146epju \u0101rstnieciskais pielietojums tiek pied\u0113v\u0113ts le\u0123end\u0101rajam \u0137\u012bnie\u0161u imperatoram \u0160e\u0146 Nunam (Shen Nung), kur\u0161, dom\u0101jams, dz\u012bvojis ap 2700. gadu p.m.\u0113. Ka\u0146epju \u0101rstniecisk\u0101 izmanto\u0161ana ir aprakst\u012bta Shen Nung Pen-ts\u2019ao Ching \u2014 2. gadsimta \u0137\u012bnie\u0161u \u0101rstniec\u012bbas augu gr\u0101mat\u0101, kur\u0101 [&#8230;]\n","protected":false},"author":1,"featured_media":2316,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[642,638,626],"tags":[633,635,634,636],"class_list":["post-2669","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-cbd","category-cbd-ellu","category-select-nekategorizetsnekategorizets","tag-cbd","tag-cbd-ella","tag-cbd-kanepju-ella","tag-sweetdropcbd"],"yoast_head":"<!-- This site is optimized with the Yoast SEO Premium plugin v27.4 (Yoast SEO v27.4) - https:\/\/yoast.com\/product\/yoast-seo-premium-wordpress\/ -->\n<title>Ka\u0146epju lieto\u0161anas medic\u012bniskie aspekti - Sweet Drop CBD<\/title>\n<meta name=\"description\" content=\"Sweet Drop CBD premium CBD oils. 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